Nutrition Specialist Exam

Section C – Supplement Topic

David Story

 

Cortislim

 

I am writing about the supplement Cortislim. I picked this supplement for my topic partially because I felt Cortislim made some inflated claims.  Midway through researching this paper it came to my attention that a lawsuit was brought up against the makers of Cortislim.  I do not know anything at all about the lawsuit.  I decided against learning more until I completed the assignment.  However, I did notice that the Cortislim website changed over the period that I wrote the paper. 

 

The most notable change on the website is the strong emphasis on the “Cortislim Lifestyle”.  The “Cortislim Lifestyle” stresses exercise, proper diet, and stress management combined with supplementation (using their product).  While these were on the website prior to the change, they were not featured as prominently on the home page as they are now.  Coinciding with this is a noticeable absence of the word cortisol on the home page, which was strongly implicated as a major barrier to weight loss.

 

Introduction:

 

The product Cortislim is billed primarily as a fat loss supplement, purportedly by controlling cortisol levels.  According to the Cortislim website, the hormone cortisol signals two actions in the body: increase of appetite and storage of fat.  While this is true, there is more to the story. 

 

Cortisol levels increase in response to stress (it is often referred to as “the stress hormone”).  Among other things, increased cortisol levels signal a breakdown of muscle tissue into amino acids to be converted into glucose by the liver (gluconeogenesis).  This allows the brain to have an uninterrupted supply of glucose under stressful conditions (1).  Cortisol performs several other jobs, like helping to maintain blood pressure and cardiovascular function, reducing the immune system’s inflammatory response, balancing the effects of insulin in breaking down sugar for energy, and regulating the metabolism of proteins, carbohydrates, and fats.

 

Normally, the production and release of cortisol is tightly controlled by the brain and pituitary & adrenal glands.  The hypothalamus sends corticotropin-releasing hormone (CRH) to the pituitary gland causing the release of adrenocorticotrophin (ACTH).  ACTH is then released into the bloodstream, acting on the adrenal glands to release cortisol. (2)

 

There is a condition, Cushing’s syndrome, in which body tissues are exposed to cortisol for prolonged periods.  It develops due to abnormal overproduction of cortisol by the adrenal glands or due to prolonged exposure of the body’s tissues to cortisol (from ingestion of corticosteroids or from tumors affecting the pituitary or adrenal glands).  Symptoms of Cushing’s syndrome include hypertension, diabetes, abdominal stretch marks, and accentuated fatty tissue on face and upper back (1).  The Cortislim website does not mention Cushing’s syndrome.

 

Theory behind cortislim:

 

Excess cortisol has been associated with an increase in appetite.  In addition, there is a pattern of fat distribution associated with excess cortisol: fat tends to be stored in the abdominal area as opposed to the hips (1).

 

Viewing the Cortislim website prior to its recent changes, it appeared Cortislim is formulated to counteract these two effects of cortisol, as well as several other mechanisms for weight loss.  These include “help balance blood sugars”, “help optimize overall metabolic rate” and “burn fat”.  Other benefits of taking Cortislim are “less stress”, “more energy”, and “better mental focus”.

 

Cortislim is composed of a number of ingredients including Calcium, Vitamin C, Chromium, and three proprietary herbal blends.  The blends are described below, followed by an explanation of their purported effect.  These explanations no longer appear on the website.

 

“Cortiplex” = Magnolia Bark Extract (1.5% honokiol) + Beta-Sitosterol + Suntheanine (100% L-Theanine)

Controls cortisol levels (to reduce fat storage and promote fat mobilization)

 

“Leptiplex” = Green Tea Extract (50% EGCG) + Bitter Orange Peel Extract (5% Synephrine)

Helps to naturally control appetite, increase energy levels and stimulate metabolism

 

“Insutrol” = Banaba Leaf extract (1% corosolic acid) + 5% Vanadyl Sulfate (5 mcg vanadium)

Helps to maintain healthy glucose levels.  Also helps to reduce cravings.

 

The remaining ingredients are gelatin, microcrystalline cellulose, water, silicon dioxide, and magnesium stearate.

 

 

Research Summary:

 

Excess Cortisol and body fat:

 

The link between excess cortisol and body fat is frequently written about in fitness and weight loss articles.  Cortisol is mentioned in the same breath as sleep deprivation, over-training, job stress or another stressor.  Readers are then admonished that the stressor (associated with the elevated cortisol) could be sabotaging their weight loss efforts, or worse, making them fat.

 

The evidence supporting these ideas has been building for years.  A study in the Annals of the New York Academy of Sciences (December 1995) showed that high cortisol levels associated with chronic stress might exert a fat storing effect on the body, particularly with regards to intra-abdominal fat (3).  Psychosomatic Medicine (the journal of the American Psychosomatic Society) published a study in February 2000 in which fifty-nine healthy pre-menopausal women were enrolled.  The women were grouped according to low (n=29) or high (n=30) WHR (Waist Hip Ratio).  A low WHR corresponded to low abdominal fat storage. The authors concluded that cortisol secretion might contribute to central fat in otherwise lean women (4). They suggested however, that excess cortisol might not be as strongly related to abdominal fat in women who are overweight.  Also, the findings cannot necessarily be applied to men, since only women were enrolled in the study.

 

Researchers at Boston’s Beth Israel Hospital and the University of Edinburgh conducted a joint animal study in 2001.  Aware that obese individuals do not typically have increased blood cortisol levels, the researchers focused on the activity of the enzyme 11beta hydroxysteroid dehydrogenase type 1 (11 beta HSD-1).  Known to be present in fat cells, 11 beta HSD-1 has the unique ability to produce cortisol in cells not normally associated with cortisol production.  The increased activity of 11 beta HSD-1 led to elevated cortisol production in fat cells, leading researchers to conclude that it might have a strong impact on abdominal obesity (5). 

 

 

Lowering excess cortisol:

 

Depending on the cause, there are a number of options for lowering excess cortisol without the use of supplements, drugs or other substances.  The choice may depend on the reason for the cortisol elevation.  More sleep, relaxation or stress management techniques, reduced intake of cortisol-elevating substances (such as caffeine), removal of a stressor and proper fitness training are all methods commonly recommended for lowering elevated cortisol levels (1).

 

Lowering cortisol in Cushing’s patients:

According to the National Institute of Diabetes and Digestive Kidney Diseases (NIDDK), there are a variety of approaches to treating Cushing’s patients.  If a tumor is the cause of the increased cortisol production, methods such as surgery, radiation, or chemotherapy are used.  If the cause is long-term use of glucocorticoid hormones to treat another disorder, a gradual dosage reduction to the lowest dose adequate for control of that disorder may be attempted.  Cortisol-inhibiting drugs are sometimes an option also (10).  Notably, it does not look as if any of the “Cortiplex” ingredients (magnolia bark, beta-sitosterol, or theanine) make up any of these cortisol-inhibiting drugs.

 

I could not find any studies or research demonstrating the cortisol lowering effects of Cortislim (my opinion on this fact follows in the “Opinion” section).  Therefore I will discuss research on the three ingredients in “Cortiplex”, the proprietary herbal blend in Cortislim stated to be responsible for lowering cortisol.  Again “Cortiplex” is made up of Magnolia Bark, Beta Sitosterol and Theanine.

 

Magnolia Bark

Magnolia bark is a traditional Chinese medicine used for treating "stagnation of qi" (low energy) as well as digestive disturbances caused by emotional distress and emotional turmoil. It is rich in magnolol and honokiol, with both compounds said to contribute to Magnolia Bark’s anti-stress and cortisol-lowering effects (6).  Animal studies have shown honokiol acts as a non-sedating, anti-anxiety and anti-stress agent at lower doses.  I was not able to find research suggesting that either honokiol or magnolol has a direct effect on cortisol or on the adrenal glands (where cortisol is produced). 

 

It looks as though the purpose of including Magnolia bark in Cortislim is to keep stress levels at bay, which would presumably influence cortisol production. The SupplementWatch website says newer claims are emerging to link magnolia bark’s anti-stress benefits with control of cortisol.  There is no evidence in the form of human studies however.

 

Beta Sitosterol

Beta-Sitosterol is a phytosterol, which is a plant compound that has a chemical structure similar to cholesterol (7).  It is sometimes used to treat prostate problems, urinary difficulties and high cholesterol.  The May 1999 International Journal of Sports Medicine published a pilot study in which nine marathoners received a supplement capsule containing Beta-Sitosterol, and eight other marathoners received a placebo.  It was determined that the Beta-Sitosterol significantly decreased the ratio of cortisol to DHEA (8).  With other effects, this was interpreted to mean Beta-Sitosterol could help lower immunosuppression responses related to exercise stress.

 

Theanine

Theanine is an amino acid found in green tea leaves.  It is thought to act as a non-sedating relaxant that helps increase the brain's production of alpha waves (brain waves associated with "relaxed alertness"). By doing so, theanine is thought to control anxiety, increase mental focus, and improve concentration (6).  In its description of L-theanine, the pdrhealth website cites a trial that involved a small group of 18-22 year old women.  The trial showed a dose-dependent increased production of alpha waves in those who consumed 200 mg of L-Theanine compared to those who consumed water.  It was suggested that more rigorous follow-up is required (9).

 

 

Controlling appetite:

 

Cortislim’s proprietary herbal blend “Leptiplex” is composed of green leaf tea extract (with EGCG) and Bitter Orange Peel Extract (with Synephrine).  Leptiplex is supposed to naturally control appetite, increase energy levels and stimulate metabolism.

 

Green Tea Leaf Extract (with EGCG)

The list of benefits attributed to green tea consumption, such as boosting the immune system and arthritis prevention, has been growing in recent years.  EGCG is one of four major catechins (polyphenols), the active components of green tea.  Antioxidant benefits ascribed to green leaf tea extract include cancer prevention, lowering of cholesterol, and reduction of blood pressure (9).  It is usually the EGCG component of green tea that is credited with contributing to appetite suppression and enhanced metabolism. 

 

In 2000, researchers at the University of Chicago's Tang Center for Herbal Medicine Research showed rats ate 50-60% less food after receiving 7 days of EGCG injections, resulting in lower body weights (11). Abdominal and subcutaneous fat, blood lipid levels, blood glucose and cholesterol all went down as well.

 

The website for “Science a GoGo” describes a study in which ten young obese males consumed green tea extract (with caffeine), caffeine alone, or placebo with a prepared meal.  Green tea consumption led to a 4% increase in thermogenesis and a 4.5% increase in overall energy expenditure. (12). The subjects that had caffeine only showed no change in metabolic rate.  The website made no reference to the study appearing in any medical or science journals.

 

A study at Shizuoka University in Japan fed 1 – 4% green tea powder to female mice for 16 weeks.  The 2% and 4% green tea powder caused a decrease of body weight, body fat and intraperitoneal (abdominal) adipose tissue.  Food intake was reduced by the 4% solution (13).   In addition, levels of cholesterol and triglycerides were lower in mice receiving the green tea diet.

 

 

Bitter Orange Peel Extract / Synephrine

A compound called octopamine, found in bitter orange peel extract, is reported to be potentially involved in appetite control.  According to chasefreedom.com, a website aimed to provide diet reviews and information, this assertion stems from a study showing that octopamine stopped bugs from eating citrus fruit (14).  However, I was unable to find evidence this study, or of any evidence of an appetite suppression effect from octopamine.

 

Synephrine is chemically similar to ephedrine, a stimulant that has gotten press for having been pulled off the market for its health risks.  Touted as a mild stimulant, synephrine is alleged to cause an elevation in metabolic rate (caloric expenditure), without the same negative cardiovascular side effects as ephedrine (6).  Synephrine is said to target some body tissues more selectively (fat cells more, heart cells less) than epinephrine.  I was unable to find research showing that synephrine is proven safe or that synephrine has an appetite suppressing effect.

 

Maintain healthy glucose levels:

“Insutrol” is composed of banaba leaf extract and vanadyl sulfate.  These are each reported to help lower blood glucose levels.

 

Banaba Leaf Extract (with 1% corosolic acid)

Banaba leaf extract is used in the Philippines to treat diabetes mellitus (15).  Corosolic acid, the active ingredient in banaba leaf, has been reported to activate glucose transport in cell cultures and to lower glucose in diabetic mice. Some reports that corosolic acid lowers blood glucose levels in type 2 diabetic subjects exist, but none of the reports has appeared in peer-reviewed scientific literature.  Additional claims for corosolic acid include burns fat, lowers elevated blood pressure and boosts energy.  According to pdrhealth.com there is “no credible evidence to support any claim for the use of corosolic acid in humans” (16).

 

Vanadyl Sulfate

Vanadyl sulfate is the most common supplemental form of a mineral called vanadium.  Vanadium is thought to imitate the effects of insulin, thus maintain blood glucose levels (6).  One study showed large doses of vanadyl sulfate lowered blood sugar levels in people with Type II diabetes, but not dramatically, according to the Nutrition Action Letter (17).  Human research on the effect of vanadium as it relates to blood glucose is scant. 

 

 

Chromium, calcium, and Vitamin C are in Cortislim as well.  There is evidence that these may have the effects that are credited to the herbal ingredients described above. These three essential nutrients are each widely consumed in supplement form.

 

Chromium

According to the UC Berkeley wellness letter, chromium is an essential mineral, but deficiency is rare in the U.S.  It plays a role in processing carbohydrates and fats, and it helps cells respond properly to insulin. It might help people with Type 2 diabetes, though this is speculative (18).

 

Calcium

Some studies have indicated that higher calcium intakes correlate with lower body fat storage.  A study of 321 girls aged nine to 14 found that those girls who consumed more calcium weighed less and had less body fat than girls who consumed the same amount of calories with less calcium.   Girls with similar calorie intake, physical activity level, and size were compared (19).

 

In another study, mice were fed a calorie-restricted diet and consumed calcium in one of three ways: a calcium supplement, a medium amount of low fat milk, or a high amount of low fat milk.  The percent fat loss for each group was 42%, 60% and 69% respectively, compared to an 8% fat loss for a group that had no calcium supplementation (20).

 

Vitamin C

A Vitamin C study demonstrated a stress reducing effect in people who were put into a stress-inducing situation.  Sixty of 120 subjects were given 1,000 mg of Vitamin C, and sixty were given placebo.  Blood pressure, cortisol, and subjective responses to a stress test were all lower in the Vitamin C group (21).

 

A 1999 rat study showed large Vitamin C doses lowered blood cortisol levels.  The doses were the equivalent of several thousand milligrams in humans. In addition, other markers of emotional and physical stress, such as body weight and enlarged adrenal glands, were positively affected (22).

 

 

References:

 

1.About.com

2.Medicinenet.com/stress

3.PUBMED -- >Peeke PM, Chrousos GP. (1995). Hypercortisolism and obesity.  Annals of the New York Academy of Sciences, 771, 665-676

4.Psychosomatic Medicine (the journal of the American Psychosomatic Society) Epel, E.S., McEwen, B., Seeman, T., Matthews, K., Castellazzo, G., Brownell, K.D., Bell, J., & Ickovics, J.R. (2000). Stress and body shape: stress-induced cortisol secretion is consistently greater among women with central fat. Psychosomatic Medicine, 62, 623-632

http://www.psychosomaticmedicine.org/cgi/content/full/62/5/623

5.http://home.caregroup.org/newsnow/pr_out.asp?pr_id=253

6.http://www.supplementwatch.com/

7.http://www.wholehealthmd.com/refshelf/substances_view/1,1525,972,00.html

8.PubMed -àInt J Sports Med. 1999 May;20(4):258-62.

9.http://www.pdrhealth.com/drug_info/nmdrugprofiles/nutsupdrugs/lth_0296.shtml

10. http://www.niddk.nih.gov/health/endo/pubs/cushings/cushings.htm

11. Endocrinology Vol. 141, No. 3 900-987. http://endo.endojournals.org/cgi/content/full/141/3/980      

12. http://scienceagogo.com/news/19991029004721data_trunc_sys.shtml

13. PubMed -à In Vivo. 2000 Jul-Aug;14(4):481-4

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=10945161&dopt=Abstract

14. chasefreedom.com

15.  http://banabaherb.com/

16.  http://www.pdrhealth.com/drug_info/nmdrugprofiles/nutsupdrugs/col_0081.shtml

17. http://www.cspinet.org/nah/05_01/

18. http://www.berkeleywellness.com/html/ds/dsChromium.php

19. http://content.health.msn.com/content/article/63/72079.htm

20. http://my.webmd.com/content/article/23/1728_56703

21. Psychopharmacology (Berl). 2002 Jan;159(3):319-24. Epub 2001 Nov 20. (PubMed)

22. http://www.anomalous-images.com/news/news499.html

 

 


Opinion:

 

Basis for product need

Based on the product name, as well as statements on their radio advertisements and website, the manufacturers of Cortislim primary aim is to implicate the hormone cortisol in people’s failure to lose weight.  While research indicates a connection between abdominal body fat and cortisol, it does not look to be a direct cause and effect scenario. Many of the studies are on animals. 

 

The study I referred to (from Psychosomatic Medicine) was a small, case control study.  The authors suggested that cortisol might not be as much of a factor for abdominal fat storage in overweight women as in lean women.  This suggests elevated cortisol can affect people differently, causing only some to store fat (the research saying cortisol has direct effect on fat deposition is inconsistent).  Also, people with high stress do not necessarily have high cortisol levels. 

 

As I write in the section on Cortislim’s marketing (below), no one would conclude such distinctions exist when looking at Cortislim’s website.  Instead there were blanket insinuations that stress leads to elevated cortisol levels which leads to weight gain and/or failure to lose weight.

 

If a client truly had elevated cortisol levels (known by getting an adrenal stress test), I’d suggest to that individual possibly more testing and definitely talking to a doctor.   In the interim, I’d recommend behavioral changes to lower cortisol levels.  More importantly, in my role as a personal trainer, I would focus on exercise as a means for combating stress and losing weight.

 

No Clinical Trial

Ideally, a double blind, placebo controlled trial would be conducted to determine the safety and efficacy of Cortislim.  A significant number of overweight subjects with high cortisol levels would need to be recruited.  Baseline cortisol and body fat percentages would need to be established for each subject.  Subjects would take Cortislim or placebo for a period, and then cortisol levels and body fat percentage would need to be measured for a second time.

 

The study would need to determine whether those who take Cortislim have lower cortisol levels and lower levels of body fat at the end of the study.  Those who took placebo would act as control group, with variables like activity levels, food intake, sleep and stress levels being controlled for also.  In addition, safety would have to be monitored. The fact that there is no such research on the safety or effectiveness of this product is the most critical reason why I am against it.  Simply put, its effects are unknown.

 

The website actually promotes undertaking lifestyle changes, like exercise, proper nutrition, and stress management, to go along with supplementation, as “a vital link to better managing your everyday stress”.

 

The suggested eating habits (in the website’s “User Guide”) include:

 

-          Eat fresh and natural whole foods. Avoid processed, artificial foods.

-          Avoid caffeine and sugar.

-          Stop eating past 7pm, or three hours before bedtime. Instead of having one large meal, break up your meals into smaller portions spread throughout the day.

-          Drink plenty of water and replace soda with water. Water suppresses appetite and helps metabolize fat. On average, a person should drink at least 8 glasses of water a day.

 

Suggested changes for managing stress include:

 

-          Take 30 minute breaks to relax

-          Get eight hours of sleep

-          Avoid stimulants like caffeine

-          Do low impact exercise

 

While these recommendations are positive, they make it impossible to know the effect of Cortislim on stress and weight management.  If the user loses weight, it may be a direct result of the lifestyle changes.  Instead of striving to isolate the effects of their product, the makers muddle the picture by encouraging consumers to use Cortislim in combination with demonstrated weight loss and stress management solutions.

 

Ingredients

Beyond the fact that there is no published research on Cortislim’s product, there does not seem to be sufficient research to support the claims for the proprietary ingredients.  Given the number of ingredients in these herbal blends (seven total), one would hope for more quality human trials to refer to.

 

The FDA monitors drug studies to ensure that they are conducted properly.  We do not have that assurance (or the assurance that there was human testing done at all) when it comes to the herbal ingredients.  Thus the safety of Cortislim is unknown.

 

In terms of efficacy, there is nothing that convinced me that Cortislim’s proprietary herbal blends has a direct effect on cortisol or on the adrenal glands’ production of cortisol.  “Cortiplex”, the blend of three herbs purportedly responsible for such an effect, at best has a calming effect that may influence anxiety levels.

 

The most promising herbal ingredient in Cortislim is green tea extract (part of “Leptiplex”.  The evidence to support the claims of appetite suppression and increased metabolism is not overly compelling, but it better than for any of other the herbal ingredient claims.  Evidence that bitter orange (with synephrine) has an appetite-suppressing effect could not be found.  While synephrine may have metabolism increasing effects, it is not clear that synephrine is necessarily safe.

 

In my opinion, the most compelling support for Cortislim’s efficacy claims can be credited to calcium and Vitamin C.  The research behind calcium’s fat loss effects and behind Vitamin C’s cortisol controlling effects is more persuasive than that of “Cortiplex” or “Leptiplex”

 

The marketing

As I said at beginning of the paper, the Cortislim website has recently changed.  The following statements were copied from the website prior to the changes:

 

·          “Anybody who leads a stressful lifestyle and wants to lose weight can benefit from CortiSlim™.  CortiSlim™ is formulated to promote weight loss, increase energy levels, and control appetite in the millions of Americans who experience stress on a daily basis. This makes CortiSlim™ the perfect product for everyone from athletes, to executives, to soccer moms, and everyone in between.”

·          CortiSlim™ should be taken as long as you have everyday stress in your life, and as long as you want to manage your weight.  If you stop taking CortiSlim™, but still have stress in your life, your cortisol levels will shoot back up, and the whole fat-making process will start again. Even after you reach your weight loss goals, you will still want to take CortiSlim™ everyday simply because of how healthy it makes you feel!

·           “Suddenly, you'll realize that your clothes are fitting more loosely, even before you've lost a single pound!”

·          CortiSlim™ will send you strong signals to avoid reaching for snacks or overeating, but it's up to you to listen. With CortiSlim™, it's easier to resist jelly donuts in the morning and a bag of chips in the afternoon. You'll realize that you will eat until you're full, instead of finishing everything on your plate. Instead of craving junk food, you'll start craving healthy foods. When stress and cortisol are no longer a controlling part of your life, you'll find freedom from food, so you'll be free to live your life!”

 

Before the changes, the website contained many misleading statements implying that virtually everyone living in our society is exposed to stress levels that will lead to increased cortisol levels.  Also, cortisol was said to be “one of the primary physiological signals for weight gain”.  Noticeably absent from the website is mention of side effects.  There is only a statement that “there will be a range of effects experienced by users”.

 

The overall content of the website solidifies my belief that Cortislim’s claims cannot be believed.  I would not recommend use of Cortislim because I doubt it’s effectiveness, and I would urge anyone who was using it to stop doing so based on the fact that its safety is unproven.